Mavoglurant racemate
Modify Date: 2024-01-06 19:10:10
Mavoglurant racemate structure
|
Common Name | Mavoglurant racemate | ||
|---|---|---|---|---|
| CAS Number | 1636881-61-2 | Molecular Weight | 313.391 | |
| Density | 1.2±0.1 g/cm3 | Boiling Point | 476.3±45.0 °C at 760 mmHg | |
| Molecular Formula | C19H23NO3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 241.8±28.7 °C | |
Use of Mavoglurant racemateMavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. |
| Name | Mavoglurant racemate |
|---|---|
| Synonym | More Synonyms |
| Description | Mavoglurant (racemate) is the racemate of mavoglurant. Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. |
|---|---|
| Related Catalog | |
| In Vitro | For antagonistic activity, (−)-mavoglurant, the (−)-enantiomer shows IC50 of 0.11 μM and 0.03 μM (Ca2+ and PI-turnover) whereas the (+)-enantiomer ((+)-10) shows only 37% and 18% inhibition at 10 μM[1]. |
| References |
| Density | 1.2±0.1 g/cm3 |
|---|---|
| Boiling Point | 476.3±45.0 °C at 760 mmHg |
| Molecular Formula | C19H23NO3 |
| Molecular Weight | 313.391 |
| Flash Point | 241.8±28.7 °C |
| Exact Mass | 313.167786 |
| LogP | 3.51 |
| Vapour Pressure | 0.0±1.3 mmHg at 25°C |
| Index of Refraction | 1.602 |
| Storage condition | 2-8℃ |
| Methyl (3aR,4S,7aR)-4-hydroxy-4-[(3-methylphenyl)ethynyl]octahydro-1H-indole-1-carboxylate |
| AFQ-056 |
| Mavoglurant |
| MFCD18633263 |
| UNII:GT0I9SV4F6 |
| 1H-Indole-1-carboxylic acid, octahydro-4-hydroxy-4-[2-(3-methylphenyl)ethynyl]-, methyl ester, (3aR,4S,7aR)- |
| Mavoglurant (racemate) |