M871
Modify Date: 2025-08-20 10:55:48
M871 structure
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Common Name | M871 | ||
|---|---|---|---|---|
| CAS Number | 908844-75-7 | Molecular Weight | 2287.61 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C108H163N27O28 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of M871M871 (Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide) is a selective galanin receptor type 2 (GalR2) antagonist. M871 exhibits Ki values of 13.1 nM and 420 nM for GalR2 and GalR1, respectively. M871 can be used for research on GalR2-related diseases (such as epilepsy, pain)[1]. |
| Name | m871 |
|---|---|
| Synonym | More Synonyms |
| Description | M871 (Galanin-(2-13)-Glu-His-(Pro)3-(Ala-Leu)2-Ala-amide) is a selective galanin receptor type 2 (GalR2) antagonist. M871 exhibits Ki values of 13.1 nM and 420 nM for GalR2 and GalR1, respectively. M871 can be used for research on GalR2-related diseases (such as epilepsy, pain)[1]. |
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| Related Catalog | |
| Target |
GalR2[1]. |
| References |
| Molecular Formula | C108H163N27O28 |
|---|---|
| Molecular Weight | 2287.61 |
| Exact Mass | 2286.22000 |
| PSA | 830.60000 |
| LogP | 2.82670 |
| InChIKey | BHKXASDHGWBINL-ZEHYZEGSSA-N |
| SMILES | CC(C)CC(NC(=O)C(C)NC(=O)C(CC(C)C)NC(=O)C(C)NC(=O)C1CCCN1C(=O)C1CCCN1C(=O)C1CCCN1C(=O)C(Cc1c[nH]cn1)NC(=O)C(CCC(=O)O)NC(=O)C1CCCN1C(=O)CNC(=O)C(CC(C)C)NC(=O)C(CC(C)C)NC(=O)C(Cc1ccc(O)cc1)NC(=O)CNC(=O)C(C)NC(=O)C(CO)NC(=O)C(CC(N)=O)NC(=O)C(CC(C)C)NC(=O)C(NC(=O)C(N)Cc1c[nH]c2ccccc12)C(C)O)C(=O)NC(C)C(N)=O |
| Storage condition | -20°C |
| trp-thr-leu-asn-ser-ala-gly-tyr-leu-leu-gly-pro-glu-his-pro-pro-pro-ala-leu-ala-leu-ala-nh2 |