Galectin-3 antagonist 1

Modify Date: 2025-08-24 22:24:49

Galectin-3 antagonist 1 Structure
Galectin-3 antagonist 1 structure
Common Name Galectin-3 antagonist 1
CAS Number 2921603-03-2 Molecular Weight 495.86
Density N/A Boiling Point N/A
Molecular Formula C22H22ClNO10 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Galectin-3 antagonist 1


Galectin-3 antagonist 1 (compound 15) is a potent and selective Galectin-3 (Gal-3) antagonist with Kd value of 5.3 μM. Meanwhile, Galectin-3 antagonist 1 binds to various Galectin with Kd values of 250 μM (Gal-4N), 18 μM (Gal-4C), 450 μM (Gal-8C), respectively[1].

 Names

Name Galectin-3 antagonist 1

 Galectin-3 antagonist 1 Biological Activity

Description Galectin-3 antagonist 1 (compound 15) is a potent and selective Galectin-3 (Gal-3) antagonist with Kd value of 5.3 μM. Meanwhile, Galectin-3 antagonist 1 binds to various Galectin with Kd values of 250 μM (Gal-4N), 18 μM (Gal-4C), 450 μM (Gal-8C), respectively[1].
Related Catalog
Target

Kd: 5.3 μM (Gal-3), 250 μM (Gal-4N), 18 μM (Gal-4C), 450 μM (Gal-8C)[1]

References

[1]. Bum-Erdene K, et al. Novel Selective Galectin-3 Antagonists Are Cytotoxic to Acute Lymphoblastic Leukemia. J Med Chem. 2022 Apr 28;65(8):5975-5989.  

 Chemical & Physical Properties

Molecular Formula C22H22ClNO10
Molecular Weight 495.86
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.