YAP-TEAD-IN-3 structure
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Common Name | YAP-TEAD-IN-3 | ||
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CAS Number | 2714434-21-4 | Molecular Weight | 529.96 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C27H26ClF2N3O4 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of YAP-TEAD-IN-3YAP-TEAD-IN-3 (compound 155) is a YAP/TAZ-TEAD inhibitor. YAP-TEAD-IN-3 inhibits Avi-humanTEAD4217-434 with an IC50 value of 9 nM. YAP-TEAD-IN-3 also inhibits NCI-H2052 with an GI50 of 0.048 μM (cell proliferation),and an IC50 of 0.048 μM (YAP reporter gene expression),respsectively[1]. |
Name | YAP-TEAD-IN-3 |
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Description | YAP-TEAD-IN-3 (compound 155) is a YAP/TAZ-TEAD inhibitor. YAP-TEAD-IN-3 inhibits Avi-humanTEAD4217-434 with an IC50 value of 9 nM. YAP-TEAD-IN-3 also inhibits NCI-H2052 with an GI50 of 0.048 μM (cell proliferation),and an IC50 of 0.048 μM (YAP reporter gene expression),respsectively[1]. |
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Related Catalog | |
Target |
IC50: 9 nM (YAP-TEAD)[1] |
References |
Molecular Formula | C27H26ClF2N3O4 |
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Molecular Weight | 529.96 |