Y08284
Modify Date: 2025-08-27 18:52:58
Y08284 structure
|
Common Name | Y08284 | ||
|---|---|---|---|---|
| CAS Number | 2688745-47-1 | Molecular Weight | 476.50 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C26H25FN4O4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Y08284Y08284 is a potent, selective, oral active CBP bromodomain inhibitor with an IC50 of 4.21 nM. Y08284 suppresses the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1. Antitumor activity[1]. |
| Name | Y08284 |
|---|
| Description | Y08284 is a potent, selective, oral active CBP bromodomain inhibitor with an IC50 of 4.21 nM. Y08284 suppresses the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1. Antitumor activity[1]. |
|---|---|
| Related Catalog | |
| In Vivo | Y08284 demonstrates favorable cell permeability and good pharmacokinetic properties, with oral bioavailability of 25.9%[1]. |
| References |
| Molecular Formula | C26H25FN4O4 |
|---|---|
| Molecular Weight | 476.50 |
| InChIKey | KKCORLIQMAQULG-UHFFFAOYSA-N |
| SMILES | COc1ccn2c(C(C)=O)cc(C(=O)Nc3cc(C(C)O)cc(-c4cnn(C5CC5)c4)c3F)c2c1 |