2688745-47-1
2688745-47-1 structure
- Name: Y08284
- Chemical Name: Y08284
- CAS Number: 2688745-47-1
- Molecular Formula: C26H25FN4O4
- Molecular Weight: 476.50
- Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
- Create Date: 2022-04-07 16:12:43
- Modify Date: 2024-01-14 09:33:31
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Y08284 is a potent, selective, oral active CBP bromodomain inhibitor with an IC50 of 4.21 nM. Y08284 suppresses the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1. Antitumor activity[1].
| Name | Y08284 |
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| Description | Y08284 is a potent, selective, oral active CBP bromodomain inhibitor with an IC50 of 4.21 nM. Y08284 suppresses the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1. Antitumor activity[1]. |
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| Related Catalog | |
| In Vivo | Y08284 demonstrates favorable cell permeability and good pharmacokinetic properties, with oral bioavailability of 25.9%[1]. |
| References |
| Molecular Formula | C26H25FN4O4 |
|---|---|
| Molecular Weight | 476.50 |