PROTAC ERα Y537S degrader-1

Modify Date: 2024-01-09 10:51:09

PROTAC ERα Y537S degrader-1 Structure
PROTAC ERα Y537S degrader-1 structure
Common Name PROTAC ERα Y537S degrader-1
CAS Number 2667598-05-0 Molecular Weight 767.91
Density N/A Boiling Point N/A
Molecular Formula C46H49N5O6 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PROTAC ERα Y537S degrader-1


PROTAC ERα Y537S degrader-1 comprises a ubiquitin E3 ligase binding group, a linker and a protein binding group. PROTAC ERα Y537S degrader-1 extracts from patent WO2021143822, example 12. PROTAC ERα Y537S degrader-1 is an estrogen receptor-alpha (ERα) Y537S degrader[1].

 Names

Name PROTAC ERα Y537S degrader-1

 PROTAC ERα Y537S degrader-1 Biological Activity

Description PROTAC ERα Y537S degrader-1 comprises a ubiquitin E3 ligase binding group, a linker and a protein binding group. PROTAC ERα Y537S degrader-1 extracts from patent WO2021143822, example 12. PROTAC ERα Y537S degrader-1 is an estrogen receptor-alpha (ERα) Y537S degrader[1].
Related Catalog
References

[1]. Yang FL, et, al. Bicyclic imide derivative, preparation method thereof, and application thereof in medicine. WO2021143822A1.

 Chemical & Physical Properties

Molecular Formula C46H49N5O6
Molecular Weight 767.91