GRK2 Inhibitor 2

Modify Date: 2024-01-16 20:17:18

GRK2 Inhibitor 2 structure	Common Name	GRK2 Inhibitor 2
	CAS Number	2592436-21-8	Molecular Weight	332.36
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₉H₁₆N₄O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of GRK2 Inhibitor 2

GRK2 Inhibitor 2 (Compound 8h) is a GRK2 inhibitor (IC50: 19 nM). GRK2 Inhibitor 2 also inhibits Aurora-A (IC50: 137 nM). GRK2 Inhibitor 2 promotes β-AR-mediated cAMP accumulation in GRK2-overexpressed HEK293 cells. GRK2 Inhibitor 2 can be used for research of congestive heart failure (HF)[1].

Name	GRK2 Inhibitor 2

Description	GRK2 Inhibitor 2 (Compound 8h) is a GRK2 inhibitor (IC50: 19 nM). GRK2 Inhibitor 2 also inhibits Aurora-A (IC50: 137 nM). GRK2 Inhibitor 2 promotes β-AR-mediated cAMP accumulation in GRK2-overexpressed HEK293 cells. GRK2 Inhibitor 2 can be used for research of congestive heart failure (HF)[1].
Related Catalog	Research Areas >> Cardiovascular Disease
References	[1]. Xu G, et al. Hit-to-lead optimization and discovery of a potent, and orally bioavailable G protein coupled receptor kinase 2 (GRK2) inhibitor. Bioorg Med Chem Lett. 2020 Dec 1;30(23):127602.

Molecular Formula	C₁₉H₁₆N₄O₂
Molecular Weight	332.36

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GRK2 Inhibitor 2

Use of GRK2 Inhibitor 2

Names

GRK2 Inhibitor 2 Biological Activity

Chemical & Physical Properties

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.