PROTAC IRAK4 degrader-1 structure
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Common Name | PROTAC IRAK4 degrader-1 | ||
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CAS Number | 2360533-90-8 | Molecular Weight | 904.85 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C44H39F3N12O7 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of PROTAC IRAK4 degrader-1PROTAC IRAK4 degrader-1 is a PROTAC interleukin-1 receptor-associated kinase 4 (IRAK4) degrader extracted from patent US20190192668A1 Compound I-210, makes <20%, >20-50%, and >50% IRAK4 degradation at 0.01, 0.1, and 1 μM in OCI-LY-10 cells, respectively[1]. |
Name | PROTAC IRAK4 degrader-1 |
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Description | PROTAC IRAK4 degrader-1 is a PROTAC interleukin-1 receptor-associated kinase 4 (IRAK4) degrader extracted from patent US20190192668A1 Compound I-210, makes <20%, >20-50%, and >50% IRAK4 degradation at 0.01, 0.1, and 1 μM in OCI-LY-10 cells, respectively[1]. |
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Related Catalog | |
Target |
IRAK4 Cereblon |
References |
[1]. Nello Mainolfi, et al. Irak degraders and uses thereof. US20190192668A1. |
Molecular Formula | C44H39F3N12O7 |
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Molecular Weight | 904.85 |
Storage condition | -20°C |