CCG 224061

Modify Date: 2024-10-07 09:49:12

CCG 224061 Structure
CCG 224061 structure
Common Name CCG 224061
CAS Number 2055990-82-2 Molecular Weight 325.387
Density N/A Boiling Point N/A
Molecular Formula C19H20FN3O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CCG 224061


A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM; displays >30-fold selectivity over GRK5, GRK1, PKA and ROCK1.

 Names

Name CCG 224061

 CCG 224061 Biological Activity

Description A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM; displays >30-fold selectivity over GRK5, GRK1, PKA and ROCK1.
References References 1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717. View Related Products by Target GRK (GPCRK)

 Chemical & Physical Properties

Molecular Formula C19H20FN3O
Molecular Weight 325.387
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