Epanolol-d5

Modify Date: 2024-01-13 18:56:18

Epanolol-d5 Structure
Epanolol-d5 structure
Common Name Epanolol-d5
CAS Number 1794938-87-6 Molecular Weight 374.45
Density N/A Boiling Point N/A
Molecular Formula C20H18D5N3O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Epanolol-d5


Epanolol-d5 (Visacor-d5) is the deuterium labeled Epanolol. Epanolol (Visacor) is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors[1][2].

 Names

Name Epanolol-d5

 Epanolol-d5 Biological Activity

Description Epanolol-d5 (Visacor-d5) is the deuterium labeled Epanolol. Epanolol (Visacor) is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors[1][2].
Related Catalog
In Vitro Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1].
References

[1]. Russak EM, et al. Impact of Deuterium Substitution on the Pharmacokinetics of Pharmaceuticals. Ann Pharmacother. 2019;53(2):211-216.

[2]. Hosie J, et al. Pharmacokinetics of epanolol after acute and chronic oral dosing in elderly patients with stable angina pectoris. Br J Clin Pharmacol. 1990 Mar;29(3):333-7.

 Chemical & Physical Properties

Molecular Formula C20H18D5N3O4
Molecular Weight 374.45