GpTx-1 structure
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Common Name | GpTx-1 | ||
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| CAS Number | 1661050-12-9 | Molecular Weight | N/A | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C176H271N53O45S7 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of GpTx-1GpTx-1 is a potent, selective, 34-residue peptide antagonist of Nav1.7 sodium channel with IC50 of 10 nM, displays 20- and 1000- fold selectivity over NaV1.4 and NaV1.5. |
| Name | GpTx-1 |
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| Description | GpTx-1 is a potent, selective, 34-residue peptide antagonist of Nav1.7 sodium channel with IC50 of 10 nM, displays 20- and 1000- fold selectivity over NaV1.4 and NaV1.5. |
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| References | References 1. Murray JK, et al. J Med Chem. 2015 Mar 12;58(5):2299-314. 2. Deuis JR, et al. Toxins (Basel). 2016 Mar 17;8(3). pii: E78. 3. Biswas K, et al. ACS Chem Biol. 2017 Sep 15;12(9):2427-2435. View Related Products by Target Sodium Channel |
| Molecular Formula | C176H271N53O45S7 |
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