orelabrutinib

Modify Date: 2024-01-11 20:08:29

orelabrutinib Structure
orelabrutinib structure
Common Name orelabrutinib
CAS Number 1655504-04-3 Molecular Weight 427.50
Density N/A Boiling Point N/A
Molecular Formula C26H25N3O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of orelabrutinib


Orelabrutinib (ICP-022) is a potent, orally active, and irreversible Bruton's tyrosine kinase (BTK) inhibitor. Orelabrutinib has the potential for B-cell malignancies treatment[1].

 Names

Name Orelabrutinib

 orelabrutinib Biological Activity

Description Orelabrutinib (ICP-022) is a potent, orally active, and irreversible Bruton's tyrosine kinase (BTK) inhibitor. Orelabrutinib has the potential for B-cell malignancies treatment[1].
Related Catalog
References

[1]. Wei Xu, et al. Safety, Tolerability and Efficacy of Orelabrutinib, Once a Day, to Treat Chinese Patients with Relapsed or Refractory Chronic Lymphocytic Leukemia/Small Cell Leukemia. Blood (2019) 134 (Supplement_1): 4319.

 Chemical & Physical Properties

Molecular Formula C26H25N3O3
Molecular Weight 427.50