RS-5773

Modify Date: 2024-02-29 16:31:52

RS-5773 Structure
RS-5773 structure
Common Name RS-5773
CAS Number 129173-57-5 Molecular Weight 547.12900
Density N/A Boiling Point 689.5ºC at 760mmHg
Molecular Formula C27H31ClN2O4S2 Melting Point N/A
MSDS N/A Flash Point 370.8ºC

 Use of RS-5773


RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction [1].

 Names

Name [(2S,3S)-5-[2-(dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-8-(thiophen-2-ylmethyl)-2,3-dihydro-1,5-benzothiazepin-3-yl] acetate,hydrochloride

 RS-5773 Biological Activity

Description RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction [1].
Related Catalog
Target

IC50: Calcium channel[1]

References

[1]. H Shiga, et al. Antianginal effect of RS-5773, a diltiazem congener, in the methacholine-induced anginal model in rats. Jpn J Pharmacol . 1996 Dec;72(4):365-74.  

 Chemical & Physical Properties

Boiling Point 689.5ºC at 760mmHg
Molecular Formula C27H31ClN2O4S2
Molecular Weight 547.12900
Flash Point 370.8ºC
Exact Mass 546.14100
PSA 112.62000
LogP 5.88780
Vapour Pressure 7.33E-19mmHg at 25°C
The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.