KNT-127
Modify Date: 2024-01-07 12:59:01
KNT-127 structure
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Common Name | KNT-127 | ||
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| CAS Number | 1256921-89-7 | Molecular Weight | 372.468 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H24N2O2 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of KNT-127A potent, selectove δ-opioid receptor agonist with Ki of 0.16 nM, dispalys 133.5-fold and 960.5-fold selectivity over μOR and κOR respectively; significantly decreases the duration of immobility and increased the duration of swimming without influencing spontaneous locomotor activity in mice (1mg/kg, s.c.). |
| Name | KNT-127 |
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| Description | A potent, selectove δ-opioid receptor agonist with Ki of 0.16 nM, dispalys 133.5-fold and 960.5-fold selectivity over μOR and κOR respectively; significantly decreases the duration of immobility and increased the duration of swimming without influencing spontaneous locomotor activity in mice (1mg/kg, s.c.). |
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| References | References 1. Nagase H, et al. Bioorg Med Chem Lett. 2010 Nov 1;20(21):6302-5. 2. Saitoh A, et al. Behav Brain Res. 2011 Oct 1;223(2):271-9. 3. Tanahashi S, et al. Neuropharmacology. 2012 Apr;62(5-6):2057-67. View Related Products by Target Opioid Receptor |
| Molecular Formula | C24H24N2O2 |
|---|---|
| Molecular Weight | 372.468 |