Terlakiren
Modify Date: 2024-02-03 21:43:15
Terlakiren structure
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Common Name | Terlakiren | ||
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| CAS Number | 119625-78-4 | Molecular Weight | 620.80 | |
| Density | 1.205g/cm3 | Boiling Point | 908.3ºC at 760mmHg | |
| Molecular Formula | C31H48N4O7S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 503.1ºC | |
Use of TerlakirenTerlakiren (CP-80,794) is an orally active inhibitor of renin. Terlakiren inhibits the efficacy of human renin with an IC50 value of 0.7 nM. Terlakiren has potential applications in hypertension[1]. |
| Name | propan-2-yl (2R,3S)-4-cyclohexyl-2-hydroxy-3-[[(2R)-3-methylsulfanyl-2-[[(2S)-2-(morpholine-4-carbonylamino)-3-phenylpropanoyl]amino]propanoyl]amino]butanoate |
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| Synonym | More Synonyms |
| Description | Terlakiren (CP-80,794) is an orally active inhibitor of renin. Terlakiren inhibits the efficacy of human renin with an IC50 value of 0.7 nM. Terlakiren has potential applications in hypertension[1]. |
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| Related Catalog | |
| References |
| Density | 1.205g/cm3 |
|---|---|
| Boiling Point | 908.3ºC at 760mmHg |
| Molecular Formula | C31H48N4O7S |
| Molecular Weight | 620.80 |
| Flash Point | 503.1ºC |
| Exact Mass | 620.32400 |
| PSA | 171.60000 |
| LogP | 3.36560 |
| Vapour Pressure | 0mmHg at 25°C |
| Index of Refraction | 1.554 |
| Terlakiren (USAN/INN) |
| N-(Morpholin-4-Ylcarbonyl)-L-Phenylalanyl-N-[(1r,2s)-1-(Cyclohexylmethyl)-2-Hydroxy-3-(1-Methylethoxy)-3-Oxopropyl]-S-Methyl-L-Cysteinamide |
| 2ZS |
| [R-(R*,S*)]-N-(4-morpholinylcarbonyl)-L-phenylalanyl-N-[1-(cyclohexylmethyl)-2-hydroxy-3-(1-methylethoxy)-3-oxopropyl]-(S)-methyl-L-cysteineamide |
| MOR-PHE-CYM-NOR |