2118899-51-5

2118899-51-5 structure

Name: Taragarestrant
Chemical Name: Taragarestrant
CAS Number: 2118899-51-5
Molecular Formula: C₂₅H₂₅Cl₂FN₂O₂
Molecular Weight: 475.38
Catalog: Research Areas Cancer
Create Date: 2022-09-30 23:41:13
Modify Date: 2025-09-21 20:15:09
Taragarestrant (D-0502) is a potent, orally active estrogen receptor degrader. Taragarestrant has antiproliferative activity against estrogen receptor-positive breast cancer cell lines and has anticancer activity. Taragarestrant can be used for cancer research[1][2].

Name	Taragarestrant

Description	Taragarestrant (D-0502) is a potent, orally active estrogen receptor degrader. Taragarestrant has antiproliferative activity against estrogen receptor-positive breast cancer cell lines and has anticancer activity. Taragarestrant can be used for cancer research[1][2].
Related Catalog	Signaling Pathways >> Others >> Estrogen Receptor/ERR Research Areas >> Cancer
References	[1]. Lin WY, et, al. Abstract 5776: Pharmacologic and PK/PD study of D-0502: An orally bioavailable SERD with potent antitumor activity in ER-positive breast cancer cell lines and xenograft models. 2018 Jul 1;78(13):5776. [2]. WHO Drug Information. International Nonproprietary Names for Pharmaceutical

Molecular Formula	C₂₅H₂₅Cl₂FN₂O₂
Molecular Weight	475.38