Name | TbPTR1 inhibitor 1 |
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Description | TbPTR1 inhibitor 1 (compound 5d) is a potent kinetoplastid pteridine reductase 1 (PTR1) inhibitor with an IC50<0.1 nM for TbPTR1. TbPTR1 inhibitor 1 has inhibitory activity against Trypanosoma brucei (EC50=0.66 μM)[1]. |
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Related Catalog | |
Target |
IC50: <0.1 nM (TbPTR1)[1] |
References |
Molecular Formula | C22H21N7O |
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Molecular Weight | 399.45 |