1974279-29-2

1974279-29-2 structure
1974279-29-2 structure
  • Name: YX-2-115
  • Chemical Name: YX-2-115
  • CAS Number: 1974279-29-2
  • Molecular Formula: C28H37N9O3
  • Molecular Weight: 547.664
  • Create Date: 2022-08-14 11:45:45
  • Modify Date: 2024-01-13 11:51:46
  • YX-2-115 is a palbociclib derivative compound with piperazine-linker tail for PROTAC YX-2-107 synthesis, inhibits CDK6 with IC50 of 4.5 nM.

Name YX-2-115
Description YX-2-115 is a palbociclib derivative compound with piperazine-linker tail for PROTAC YX-2-107 synthesis, inhibits CDK6 with IC50 of 4.5 nM.
References 1. Marco De Dominici, et al. Blood. 2020 Apr 30;135(18):1560-1573.
Molecular Formula C28H37N9O3
Molecular Weight 547.664