2685738-33-2
2685738-33-2 structure
- Name: ER-001259851-000
- Chemical Name: ER-001259851-000
- CAS Number: 2685738-33-2
- Molecular Formula: C36H41FN8O4
- Molecular Weight: 668.774
- Create Date: 2022-07-02 07:43:34
- Modify Date: 2025-11-03 17:40:25
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ER-001259851-000 is a potent, selective, orally active Axl inhibitor with IC50 of 5.2 nM in cell free assays, displays >35-fold selectivity against Mer (IC50=190 nM).ER-001259851-000 shows a promising pharmacokinetic profile in mice.
| Name | ER-001259851-000 |
|---|
| Description | ER-001259851-000 is a potent, selective, orally active Axl inhibitor with IC50 of 5.2 nM in cell free assays, displays >35-fold selectivity against Mer (IC50=190 nM).ER-001259851-000 shows a promising pharmacokinetic profile in mice. |
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| References | 1. Satoshi Inoue, et al. Bioorg Med Chem Lett. 2021 Sep 15;48:128247. |
| Molecular Formula | C36H41FN8O4 |
|---|---|
| Molecular Weight | 668.774 |