2170126-74-4

2170126-74-4 structure

Name: BMS-986278
Chemical Name: BMS-986278
CAS Number: 2170126-74-4
Molecular Formula: C₂₂H₃₁N₅O₅
Molecular Weight: 445.51
Catalog: Signaling Pathways GPCR/G Protein LPL Receptor
Create Date: 2022-01-07 13:51:00
Modify Date: 2024-01-03 10:25:43
BMS-986278 is a potent lysophosphatidic acid receptor 1 (LPA1) antagonist, with a human LPA1 Kb of 6.9 nM.

Name	BMS-986278

Description	BMS-986278 is a potent lysophosphatidic acid receptor 1 (LPA1) antagonist, with a human LPA1 Kb of 6.9 nM.
Related Catalog	Research Areas >> Others Signaling Pathways >> GPCR/G Protein >> LPL Receptor
References	[1]. Cheng PTW, et al. Murphy BJ. Discovery of an Oxycyclohexyl Acid Lysophosphatidic Acid Receptor 1 (LPA1) Antagonist BMS-986278 for the Treatment of Pulmonary Fibrotic Diseases. J Med Chem. 2021 Nov 11;64(21):15549-15581.