- Zhejiang Hangyu API Co., Ltd
- China
- Product Name: (Ala1·3·11·15)-Endothelin-1
- Price: $Inquiry/1kg
- Purity: 99.0%
- Stocking Period: 1 Day
- Contact: Vinnie
121204-87-3
121204-87-3 structure
- Name: (Ala1.3.11.15)-Endothelin-1 trifluoroacetate salt
- Chemical Name: [Ala1,3,11,15]-Endothelin
- CAS Number: 121204-87-3
- Molecular Formula: C109H163N25O32S
- Molecular Weight: 2367.674
- Catalog: Biochemical Amino acids and their derivatives Alanine derivatives
- Create Date: 2018-06-19 23:26:08
- Modify Date: 2024-01-10 23:00:45
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[Ala1,3,11,15]-Endothelin (53-63) is an ETB agonist. [Ala1,3,11,15]-Endothelin (53-63) has selectivity for ETB with IC50 values range from 0.33 nM to 0.61 nM. [Ala1,3,11,15]-Endothelin (53-63) can be used for the research of vasoconstriction[1][2].
| Name | [Ala1,3,11,15]-Endothelin |
|---|---|
| Synonyms |
asasslmdkeavyfahldiiw
L-Tryptophan, L-alanyl-L-seryl-L-alanyl-L-seryl-L-seryl-L-leucyl-L-methionyl-L-α-aspartyl-L-lysyl-L-α-glutamyl-L-alanyl-L-valyl-L-tyrosyl-L-phenylalanyl-L-alanyl-L-histidyl-L-leucyl-L-α-as
 partyl-L-isoleucyl-L-isoleucyl- ala-ser-ala-ser-ser-leu-met-asp-lys-glu-ala-val-tyr-phe-ala-his-leu-asp-ile-ile-trp MFCD00143562 L-Alanyl-L-seryl-L-alanyl-L-seryl-L-seryl-L-leucyl-L-methionyl-L-α-aspartyl-L-lysyl-L-α-glutamyl-L-alanyl-L-valyl-L-tyrosyl-L-phenylalanyl-L-alanyl-L-histidyl-L-leucyl-L-α-aspartyl-L-isole
 ucyl-L-isoleucyl-L-tryptophan 4 ala et-1 |
| Description | [Ala1,3,11,15]-Endothelin (53-63) is an ETB agonist. [Ala1,3,11,15]-Endothelin (53-63) has selectivity for ETB with IC50 values range from 0.33 nM to 0.61 nM. [Ala1,3,11,15]-Endothelin (53-63) can be used for the research of vasoconstriction[1][2]. |
|---|---|
| Related Catalog | |
| Target |
IC50 for ETB: 0.61 nM (Bronchus); 0.61 nM (Lung); 0.33 nM (Cerebellum); 2200 nM (VSMC)[1] |
| In Vitro | [Ala1,3,11,15]-Endothelin (53-63) (0.1 μM) has selectivity for ETB with IC50 values of 0.61 nM, 0.61 nM, 0.33 nM, 2200 nM in Bronchus, Lung, Cerebellum and VSMC, respectively[1]. |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 2391.5±65.0 °C at 760 mmHg |
| Molecular Formula | C109H163N25O32S |
| Molecular Weight | 2367.674 |
| Flash Point | 1400.1±34.3 °C |
| Exact Mass | 2366.161621 |
| PSA | 933.93000 |
| LogP | 3.12 |
| Vapour Pressure | 0.0±0.3 mmHg at 25°C |
| Index of Refraction | 1.586 |
| Storage condition | −20°C |
| Personal Protective Equipment | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
|---|---|
| RIDADR | NONH for all modes of transport |
| WGK Germany | 3 |