2469274-58-4

2469274-58-4 structure
2469274-58-4 structure
  • Name: Palosuran hydrochloride
  • Chemical Name: Palosuran hydrochloride
  • CAS Number: 2469274-58-4
  • Molecular Formula: C25H31ClN4O2
  • Molecular Weight: 454.99
  • Create Date: 2021-05-31 12:41:14
  • Modify Date: 2024-02-22 09:40:11
  • Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. Palosuran hydrochloride can improves pancreatic and renal function in diabetic rats.

Name Palosuran hydrochloride
Description Palosuran hydrochloride (ACT-058362 hydrochloride) is a potent, selective, and orally active antagonist of urotensin II receptor, with an IC50 of 3.6 nM for CHO cell membranes expressing human recombinant receptors. Palosuran hydrochloride can improves pancreatic and renal function in diabetic rats.
Molecular Formula C25H31ClN4O2
Molecular Weight 454.99