Name | RVD-Hpα |
---|
Description | RVD-Hpα is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα also high affinity CB2 positive allosteric modulator (Ki=50 nM). |
---|---|
Related Catalog | |
Target |
CB1 |
Molecular Formula | C65H105N19O17 |
---|---|
Molecular Weight | 1424.66 |