| Name | RVD-Hpα |
|---|
| Description | RVD-Hpα is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα also high affinity CB2 positive allosteric modulator (Ki=50 nM). |
|---|---|
| Related Catalog | |
| Target |
CB1 |
| Molecular Formula | C65H105N19O17 |
|---|---|
| Molecular Weight | 1424.66 |