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Product Name: OMDM-4
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616884-65-2

616884-65-2 structure

616884-65-2 structure

Name: OMDM-4
Chemical Name: OMDM-4
CAS Number: 616884-65-2
Molecular Formula: C₂₉H₄₃NO₃
Molecular Weight: 453.66
Catalog: Research Areas Neurological Disease
Create Date: 2020-06-01 21:26:28
Modify Date: 2024-01-26 07:24:27
OMDM-4 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki 17.7 μM[1].

Name	OMDM-4

Description	OMDM-4 is a selective and metabolically stable inhibitor of anandamide cellular uptake (ACU), with a Ki 17.7 μM[1].
Related Catalog	Research Areas >> Neurological Disease
Target	Ki: 17.7 μM (anandamide cellular uptake)[1]
In Vitro	OMDM-4 shows poor affinity for either CB1 (Ki=4.9 μM) or CB2 (Ki>10 μM) receptors in rat brain and spleen membranes, respectively. OMDM-4 has almost no activity at vanilloid receptors in the intracellular calcium assay carried out with intact cells over-expressing the human VR1 (EC50>10 μM), and no activity as inhibitors of FAAH in N18TG2 cell membranes (Ki>50 μM)[1].
References	[1]. Ortar G, et al. Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem Pharmacol. 2003 May 1;65(9):1473-81.

Molecular Formula	C₂₉H₄₃NO₃
Molecular Weight	453.66

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