1378183-16-4
1378183-16-4 structure
- Name: ZINC-3573 racemate
- Chemical Name: ZINC-3573 racemate
- CAS Number: 1378183-16-4
- Molecular Formula: C18H21N5
- Molecular Weight: 307.401
- Create Date: 2020-01-11 22:42:49
- Modify Date: 2024-04-03 10:40:04
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ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases; activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release.
| Name | ZINC-3573 racemate |
|---|
| Description | ZINC-3573 racemate is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=3 uM), showing little activity against 315 other GPCRs and 97 representative kinases; activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release. |
|---|---|
| References | References 1. Lansu K, et al. Nat Chem Biol. 2017 May;13(5):529-536. View Related Products by Target Other Targets |
| Molecular Formula | C18H21N5 |
|---|---|
| Molecular Weight | 307.401 |