| Name | Taltirelin acetate |
|---|
| Description | Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 910 nM (Thyrotropin-releasing hormone receptor)[1] |
| References |
| Molecular Formula | C19H27N7O7 |
|---|---|
| Molecular Weight | 465.46 |