Name | Taltirelin acetate |
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Description | Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)[1]. |
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Related Catalog | |
Target |
IC50: 910 nM (Thyrotropin-releasing hormone receptor)[1] |
References |
Molecular Formula | C19H27N7O7 |
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Molecular Weight | 465.46 |