Name | ERK2 IN-1 |
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Description | ERK2 IN-1 is a selective ERK2 inhibitor with an IC50 of 7 nM[1]. |
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Related Catalog | |
Target |
ERK2:7 nM (IC50) |
In Vitro | ERK1/2 IN-1 (Compound 28) maintains good ERK enzymatic activity (ERK IC50=7 nM) and cellular activity in BRAF/KRAS mutant wildtype cancer cell lines (HT-29/Caspase IC50=118/80 nM)[1]. |
References |
Molecular Formula | C36H34FN7O2S |
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Molecular Weight | 647.76 |