391610-37-0
391610-37-0 structure
- Name: MCHr1 antagonist 1
- Chemical Name: MCHr1 antagonist 1
- CAS Number: 391610-37-0
- Molecular Formula: C28H33F2N5O5
- Molecular Weight: 557.59
- Catalog: Signaling Pathways GPCR/G Protein MCHR1 (GPR24)
- Create Date: 2018-05-05 05:34:53
- Modify Date: 2025-08-26 16:56:04
-
MCHr1 antagonist 1 is a selective antagonist of melanin concentrating hormone-1 (MCH1) receptor, with a Kb of 1 nM and a Ki of 4 nM at human MCH1, and may be used to reduce the body mass.
| Name | MCHr1 antagonist 1 |
|---|
| Description | MCHr1 antagonist 1 is a selective antagonist of melanin concentrating hormone-1 (MCH1) receptor, with a Kb of 1 nM and a Ki of 4 nM at human MCH1, and may be used to reduce the body mass. |
|---|---|
| Related Catalog | |
| Target |
Kb: 1 nM (Human MCH1)[1] Ki: 4 nM (Human MCH1)[1] |
| In Vitro | MCHr1 antagonist 1 shows potent activities against melanin concentrating hormone-1 receptor, but less potent against human MCH1, NPY1, NPY5, GALR1, GALR2, GALR3, and rat 5HT2C receptors, with Kis of >50000 nM[1]. |
| References |
| Molecular Formula | C28H33F2N5O5 |
|---|---|
| Molecular Weight | 557.59 |