Name | Cicloprolol hydrochloride |
---|---|
Synonyms |
(±)-1-(p-(2-(Cyclopropylmethoxy)ethoxy)phenoxy)-3-(isopropylamino)-2-propanol Hydrochloride
1-{4-[2-(Cyclopropylmethoxy)ethoxy]phenoxy}-3-(isopropylamino)-2-propanol hydrochloride (1:1) 2-Propanol, 1-[4-[2-(cyclopropylmethoxy)ethoxy]phenoxy]-3-[(1-methylethyl)amino]-, hydrochloride (1:1) (±)-1-(4-(2-(Cyclopropylmethoxy)ethoxy)phenoxy)-3-((1-methylethyl)amino)-2-propanol Hydrochloride cicloprolol hydrochloride sl-d 177 UNII:T355YD4791 T355YD4791 |
Description | Cicloprolol is a partial β 1-adrenoceptor agonist . |
---|---|
Related Catalog | |
Target |
Adrenoceptor[1] |
In Vitro | Cicloprolol is a partial β1-adrenoceptor agonist considered for the treatment of patients with coronary artery disease and impaired left ventricular function[1]. The new β-adrenoceptor partial agonist Cicloprolol acts as a β-agonist at normal levels and as a β-antagonist at high levels of adrenergic discharge. Treatment with Cicloprolol should protect the heart against excessive stimulation, while providing a baseline level of sympathetic drive. Cicloprolol has a weak β1-agonistic effect at normal levels of adrenergic discharge and acts as an antagonist at high levels of discharge[2]. |
References |
Molecular Formula | C18H30ClNO4 |
---|---|
Molecular Weight | 359.888 |
Exact Mass | 359.186340 |