EP1-antanoist-1

Names

[ CAS No. ]:
851204-35-8

[ Name ]:
EP1-antanoist-1

Biological Activity

[Description]:

EP1-antanoist-1 is a EP1 antagonist with a pKi of 7.54 and an pIC50 of 8.5.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Prostaglandin Receptor

Research Areas >> Neurological Disease

[Target]

EP1:8.5 (pIC50)

EP1:7.54 (pKi)

[References]

[1]. McKeown SC, et al. Identification of novel pyrazole acid antagonists for the EP1 receptor. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4767-71. Epub 2006 Jul 14.

[Related Small Molecules]

Dinoprostone | Prostaglandin E1 | E7046 | ONO-AE3-208 | PF 04418948 | Fevipiprant | grapiprant | TG6-10-1 | Taprenepag | GW 627368 | MRE-269 | Ramatroban | AH 6809 | Laropiprant | AZD1981

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₉H₁₅BrCl₂N₂O₃

[ Molecular Weight ]:
470.14

Related Compounds

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