AP-C3

Names

[ Name ]:
AP-C3

Biological Activity

[Description]:

AP-C3 is a potent inhibitor of guanosine 3′,5′-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) with a pIC50 of 6.3. AP-C3 only weakly inhibits cGKII-dependent anion secretion[1].

[Related Catalog]:

Research Areas >> Others

Signaling Pathways >> Others >> Others

[Target]

pIC50: 6.5 (cGKII)[1]

[References]

[1]. Marcel J C Bijvelds, et al. Selective inhibition of intestinal guanosine 3',5'-cyclic monophosphate signaling by small-molecule protein kinase inhibitors. J Biol Chem. 2018 May 25;293(21):8173-8181.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₂H₂₃N₃O₄

[ Molecular Weight ]:
393.44

Related Compounds

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