AP-C4

Names

[ CAS No. ]:
682794-85-0

[ Name ]:
AP-C4

Biological Activity

[Description]:

AP-C4 is an inhibitor of guanosine 3′,5′-cyclic monophosphate (cGMP)-dependent protein kinase II (cGKII) with a pIC50 of 5.2. AP-C3 does not inhibit cGKII-dependent anion secretion[1].

[Related Catalog]:

Research Areas >> Others
Signaling Pathways >> Others >> Others

[Target]

pIC50: 5.2 (cGKII)[1]


[References]

[1]. Marcel J C Bijvelds, et al. Selective inhibition of intestinal guanosine 3',5'-cyclic monophosphate signaling by small-molecule protein kinase inhibitors. J Biol Chem. 2018 May 25;293(21):8173-8181.  

Chemical & Physical Properties

[ Molecular Formula ]:
C22H20N4O2

[ Molecular Weight ]:
372.42


Related Compounds

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