<Suppliers Price>

benzquinamide

Names

[ CAS No. ]:
63-12-7

[ Name ]:
benzquinamide

[Synonym ]:
P2647

Biological Activity

[Description]:

Benzquinamide is an antiemetic which can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) with Ki values of 1,365, 691, and 545 nM, respectively.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> Adrenergic Receptor
Research Areas >> Metabolic Disease

[Target]

Ki: 1,365 nM (α2A), 691 nM (α2B), 545 nM (α2C)[1].


[References]

[1]. Elisabet Gregori-Puigjané, et al. Identifying mechanism-of-action targets for drugs and probes. Proc Natl Acad Sci U S A. 2012 Jul 10; 109(28): 11178-11183. doi: 10.1073/pnas.1204524109


[Related Small Molecules]

Isoprenaline hydrochloride | ICI 118,551 (hydrochloride) | Phenylephrine hydrochloride | Yohimbine hydrochloride | Adrenaline | Ivabradine hydrochloride | Prazosin hydrochloride | Clenbuterol hydrochloride | Phentolamine mesilate | guanfacine hydrochloride | pimozide | Sotalol hydrochloride | Carvedilol | Atenolol | Metroprolol succinate

Chemical & Physical Properties

[ Density]:
1.2±0.1g/cm3

[ Boiling Point ]:
531.0±50.0°C at 760 mmHg

[ Molecular Formula ]:
C22H32N2O5

[ Molecular Weight ]:
404.50000

[ Flash Point ]:
274.9±30.1°C

[ Exact Mass ]:
404.23100

[ PSA ]:
68.31000

[ LogP ]:
2.36090

Related Compounds

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.