MRS2298

Names

[ Name ]:
MRS2298

[Synonym ]:
MRS 2298
MRS-2298

Biological Activity

[Description]:

MRS2298? is a potent acyclic P2Y1 receptor antagonist with a Ki of 29.6 nM. MRS2298 inhibits the ADP-induced aggregation of human platelets with an IC50 of 62.8 nM. MRS2298 inhibits Ca2+ rise in platelets with an IC50 of 810 nM[1].

[Related Catalog]:

Research Areas >> Cardiovascular Disease

Signaling Pathways >> GPCR/G Protein >> P2Y Receptor

[References]

[1]. Marco Cattaneo, et al. Antiaggregatory activity in human platelets of potent antagonists of the P2Y 1 receptor. Biochem Pharmacol. 2004 Nov 15;68(10):1995-2002.

Chemical & Physical Properties

[ Density]:
2.03±0.1 g/cm3(Predicted)

[ Boiling Point ]:
735.8±70.0 °C(Predicted)

[ Molecular Formula ]:
C₁₀H₁₆ClN₅O₈P₂

[ Molecular Weight ]:
431.66

Related Compounds

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