ARN272

Names

[ Name ]:
ARN272

[Synonym ]:
Benzamide, 4-[[4-(4-hydroxyphenyl)-1-phthalazinyl]amino]-N-phenyl-
4-{[4-(4-Hydroxyphenyl)-1-phthalazinyl]amino}-N-phenylbenzamide

Biological Activity

[Description]:

ARN272 is an anandamide transport inhibitor[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others

Research Areas >> Neurological Disease

[Target]

Anandamide transport[1]

[References]

[1]. O'Brien LD, et al. Anandamide transport inhibition by ARN272 attenuates nausea-induced behaviour in rats, and vomiting in shrews (Suncus murinus). Br J Pharmacol. 2013 Nov;170(5):1130-6.

Chemical & Physical Properties

[ Density]:
1.4±0.1 g/cm3

[ Boiling Point ]:
629.1±55.0 °C at 760 mmHg

[ Molecular Formula ]:
C₂₇H₂₀N₄O₂

[ Molecular Weight ]:
432.473

[ Flash Point ]:
334.3±31.5 °C

[ Exact Mass ]:
432.158630

[ LogP ]:
4.58

[ Vapour Pressure ]:
0.0±1.9 mmHg at 25°C

[ Index of Refraction ]:
1.757

[ Storage condition ]:
2-8℃

Related Compounds

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