RPL-554

Names

[ Name ]:
RPL-554

[Synonym ]:
unii-3e3d8t1gix
rpl-554

Biological Activity

[Description]:

(E/Z)-Ensifentrine is a dual inhibitor of PDE3/4. (E/Z)-Ensifentrine reduces the inflammatory cells into the airways. (E/Z)-Ensifentrine has bronchodilatory and anti-inflammatory activities in vitro and in vivo model[1].

[Related Catalog]:

Signaling Pathways >> Metabolic Enzyme/Protease >> Phosphodiesterase (PDE)

Research Areas >> Neurological Disease

[References]

[1]. Page CP, et al. Phosphodiesterase inhibitors for the treatment of asthma and chronic obstructive pulmonary disease. Int Arch Allergy Immunol. 2014;165(3):152-64.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₆H₃₁N₅O₄

[ Molecular Weight ]:
477.56

[ Exact Mass ]:
477.23800

[ PSA ]:
113.86000

[ LogP ]:
3.62070

Related Compounds

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