Dim16
Names
[ CAS No. ]:
2743448-32-8
[ Name ]:
Dim16
Biological Activity
[Description]:
Dim16 is a dual PCSK9/HMG-CoAR inhibitor, with an IC50 value of 19 nM for PCSK9. Dim16 inhibits PCSK9-LDLR binding with an IC50 value of 0.8 nM. Dim16 increases LDL uptake in HepG2 cells[1].
[Related Catalog]:
[Target]
19 nM (PCSK9)[1]
[References]
Chemical & Physical Properties
[ Molecular Formula ]:
C29H38IN5
[ Molecular Weight ]:
583.55