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MRGPRX1 agonist 1

Names

[ CAS No. ]:
2377379-39-8

[ Name ]:
MRGPRX1 agonist 1

Biological Activity

[Description]:

MRGPRX1 agonist 1 is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1), with an EC50 of 50 nM, and is inactive on MRGPRC11. Analgesic effect[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others

[Target]

EC50: 50 nM (MRGPRX1)[1]


[References]

[1]. Prchalová E, et al. Discovery of Benzamidine- and 1-Aminoisoquinoline-Based Human MAS-Related G-Protein-Coupled Receptor X1 (MRGPRX1) Agonists. J Med Chem. 2019 Sep 26;62(18):8631-8641.

Chemical & Physical Properties

[ Molecular Formula ]:
C23H21N3O4S

[ Molecular Weight ]:
435.50

[ Storage condition ]:
-20°C

Related Compounds