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5-HT7R antagonist 1 free base

Names

[ CAS No. ]:
2337008-64-5

[ Name ]:
5-HT7R antagonist 1 free base

Biological Activity

[Description]:

5-HT7R antagonist 1 (free base) is a G protein-biased antagonist against 5-HT7R (Ki = 6.5 nM).

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> GPCR19
Research Areas >> Neurological Disease

[References]

[1]. Kwag R, et al. Discovery of G Protein-Biased Antagonists against 5-HT7R. J Med Chem. 2021 Sep 23;64(18):13766-13779.

Chemical & Physical Properties

[ Molecular Formula ]:
C14H17ClN4

[ Molecular Weight ]:
276.76

Related Compounds