ACT-1004-1239

Names

[ CAS No. ]:
2178049-58-4

[ Name ]:
ACT-1004-1239

Biological Activity

[Description]:

ACT-1004-1239 is a potent, selective, orally available CXCR7 antagonist with an IC50 value of 3.2 nM.

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> GPCR/G Protein >> CXCR

Research Areas >> Inflammation/Immunology

Signaling Pathways >> Immunology/Inflammation >> CXCR

Research Areas >> Neurological Disease

[References]

[1]. Richard-Bildstein S, et al. Discovery of the Potent, Selective, Orally Available CXCR7 Antagonist ACT-1004-1239. J Med Chem. 2020 Dec 24;63(24):15864-15882.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₇H₂₈F₂N₆O₃

[ Molecular Weight ]:
522.55

Related Compounds

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