BMS-212
Names
[ CAS No. ]:
2173153-38-1
[ Name ]:
BMS-212
Biological Activity
[Description]:
BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic.
[In Vitro]
BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic. BMS-212 has a preference for GK in liver over GK in pancreas, of which the activation may lead to non-glucose-dependent insulin secretion. Half-life of BMS-212 is 4.2h, and oral bioavailability is 15%.
Chemical & Physical Properties
[ Molecular Formula ]:
C25H30N3O9PS2
[ Molecular Weight ]:
611.621
Related Compounds
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