LSD1-IN-11p

Names

[ CAS No. ]:
2101951-67-9

[ Name ]:
LSD1-IN-11p

Biological Activity

[Description]:

LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%).

[References]

References 1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195. View Related Products by Target Histone Demethylase

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₂H₂₄N₆O₃

[ Molecular Weight ]:
420.473

Related Compounds

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