HSL-IN-1

Names

[ CAS No. ]:
2095156-13-9

[ Name ]:
HSL-IN-1

Biological Activity

[Description]:

HSL-IN-1 (compound 24b) is a potent and orally active hormone sensitive lipase (HSL) inhibitor (IC50=2 nM) with a significantly reduced reactive metabolite liability[1].

[Related Catalog]:

Signaling Pathways >> Others >> Others

Research Areas >> Metabolic Disease

[Target]

IC50: 2 nM (Hormone sensitive lipase)[1]

[References]

[1]. Ogiyama T, et al. Identification of a novel hormone sensitive lipase inhibitor with a reduced potential of reactive metabolites formation. Bioorg Med Chem. 2017 Apr 1;25(7):2234-2243.

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₉H₁₃BClF₃N₂O₄

[ Molecular Weight ]:
436.58

Related Compounds

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