5-HT2A antagonist 1

Names

[ CAS No. ]:
204643-75-4

[ Name ]:
5-HT2A antagonist 1

Biological Activity

[Description]:

5-HT2A antagonist 1 is a 5-HT2A antagonist extracted from patent US5728835A and JP 1007727. 5-HT2A antagonist 1 may be useful in treatment of gastrointestinal disorders circulatory disorders.

[Related Catalog]:

Signaling Pathways >> GPCR/G Protein >> 5-HT Receptor
Signaling Pathways >> Neuronal Signaling >> 5-HT Receptor
Research Areas >> Cardiovascular Disease

[Target]

5-HT2A[1]


[In Vitro]

Please refer to patent US5728835A and JP 1007727 for more information[1][2].

[References]

[1]. Aoki Tsuyoshi, et al. Substituted cyclic amine compound, production process thereof and pharmaceutical composition for circulatory organ use containing the same. US5728835A

[2]. Preparation of 3-​pyridylamines as 5-​HT2 receptor antagonists for treatment of circulatory disorders


[Related Small Molecules]

Harmine | Pimavanserin | Serotonin hydrochloride | Sodium Ferulate | Thioridazine hydrochloride | Brexpiprazole | Risperidone | TG6-10-1 | Cariprazine | Quetiapine | SERTINDOLE | Alprenolol hydrochloride | B-HT 920 | Ketanserin | Palonosetron hydrochloride

Chemical & Physical Properties

[ Molecular Formula ]:
C26H28N4O2

[ Molecular Weight ]:
428.53

Related Compounds