Molibresib besylate

Names

[ CAS No. ]:
1895049-20-3

[ Name ]:
Molibresib besylate

Biological Activity

[Description]:

Molibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM.

[Related Catalog]:

Research Areas >> Cancer

Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain

[Target]

IC50: 32.5-42.5 nM (BET)[1]

[References]

[1]. Nicodeme E, et al. Suppression of inflammation by a synthetic histone mimic. Nature. 2010 Dec 23;468(7327):1119-23.

Chemical & Physical Properties

[ Molecular Formula ]:
C₂₈H₂₈ClN₅O₅S

[ Molecular Weight ]:
582.07

[ Storage condition ]:
2-8℃

Related Compounds

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