1895049-20-3

1895049-20-3 structure
1895049-20-3 structure
  • Name: Molibresib besylate
  • Chemical Name: Molibresib besylate
  • CAS Number: 1895049-20-3
  • Molecular Formula: C28H28ClN5O5S
  • Molecular Weight: 582.07
  • Catalog: Signaling Pathways Epigenetics Epigenetic Reader Domain
  • Create Date: 2019-06-24 18:59:29
  • Modify Date: 2024-01-13 14:33:44
  • Molibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM.

Name Molibresib besylate
Description Molibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM.
Related Catalog
Target

IC50: 32.5-42.5 nM (BET)[1]

References

[1]. Nicodeme E, et al. Suppression of inflammation by a synthetic histone mimic. Nature. 2010 Dec 23;468(7327):1119-23.

Molecular Formula C28H28ClN5O5S
Molecular Weight 582.07
Storage condition 2-8℃