PF-06649298

Names

[ Name ]:
PF-06649298

Biological Activity

[Description]:

PF-06649298 (PF06649298) potent, selective inhibitor of the Na+/citrate transporter NaCT (SLC13A5) that shows inhibition of citrate uptake in the HEKNaCT cells with IC50 of 0.41 uM; displays >60-fold selectvity over NaDC1 and NaDC3.

[References]

References 1. Pajor AM, et al. Mol Pharmacol. 2016 Dec;90(6):755-765. View Related Products by Target Sodium-coupled Citrate Transporter (NaCT,SLC13A5)

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₆H₂₂O₅

[ Molecular Weight ]:
294.347

Related Compounds

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