Idelalisib D5

Names

[ CAS No. ]:
1830330-31-8

[ Name ]:
Idelalisib D5

Biological Activity

[Description]:

Idelalisib D5 is a deuterium labeled Idelalisib. Idelalisib is a highly selective and orally bioavailable p110δ inhibitor[1].

[Related Catalog]:

Research Areas >> Cancer
Signaling Pathways >> PI3K/Akt/mTOR >> PI3K
Signaling Pathways >> Autophagy >> Autophagy

[Target]

P110δ inhibitor


[References]

[1]. Lannutti BJ, et al. CAL-101, a p110delta selective phosphatidylinositol-3-kinase inhibitor for the treatment of B-cell malignancies, inhibits PI3K signaling and cellular viability. Blood, 2011, 117(2), 591-594.

Chemical & Physical Properties

[ Molecular Formula ]:
C22H13D5FN7O

[ Molecular Weight ]:
420.45


Related Compounds