PSB-12553

Names

[ Name ]:
PSB-12553

Biological Activity

[Description]:

PSB-12553 is an α,β-Methylene-ADP (AOPCP) derivative, potent, selective ecto-5′-Nucleotidase (eN, CD73) inhibitor with Ki of 9.5 nM for rat recombinant eN; displays high selectivity versus other ecto-nucleotidases and ADP-activated P2Y receptors, has high metabolic stability.

[References]

References 1. Bhattarai S, et al. J Med Chem. 2015 Aug 13;58(15):6248-63. View Related Products by Target Other Targets

Chemical & Physical Properties

[ Molecular Formula ]:
C₁₈H₂₂N₄O₉P₂S

[ Molecular Weight ]:
532.401

Related Compounds

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